SCHEMBL6941874

SCHEMBL6941874

COc1cc(C(=O)NC(=O)NN[C@@H](CC(=O)O)C(N)=O)ccc1NC(=N)N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 8/20 0.42
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CHEK1 O14757 1/20 0.39
PIM1 P11309 1/20 0.39
MAPK8 P45983 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
F10 P00742 1/20 0.38
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
EPHX1 P07099 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6934969 0.78 ITGB3 (0.51) NPC1RAB9ACHEK1PIM1MAPK8
SCHEMBL6941352 0.77 ITGB3 (0.47) F10
SCHEMBL6935372 0.75 NPC1 (0.38) NPC1RAB9AF10
SCHEMBL7879691 0.72 ITGB3 (0.56) NPC1RAB9ACHEK1PIM1MAPK8
Hydrochloric Acid SCHEMBL31158180 0.71 PYGL (0.54) PYGLNPC1RAB9AF10KMT2A
SCHEMBL6937428 0.65 ITGB3 (0.40)
SCHEMBL6935740 0.65 ITGB3 (0.46) NPC1RAB9ACHEK1PIM1MAPK8
SCHEMBL31104220 0.65 PYGL (0.57) PYGLNPC1RAB9ACHEK1PIM1
SCHEMBL7882801 0.65 ALDH1A1 (0.41) ALDH1A1
SCHEMBL7879657 0.65 ABCC1 (0.39) PYGLKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US claimed
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed