SCHEMBL6944461

SCHEMBL6944461

Nc1ncc2nc(Cc3cccnc3)[nH]c2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40
PNP P00491 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
MPO P05164 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
MMP2 P08253 1/20 0.38
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CHRNA7 P36544 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
CHRNB2 P17787 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946589 0.85 MAPT (0.37) CACNA1HHRH4HRH3CYP1A2CYP2D6
SCHEMBL6947942 0.80 EGFR (0.43) MPOCYP1A2CYP2D6GAAKDM4E
SCHEMBL6939915 0.79 DHFR (0.56) KMT2ACYP1A2GAAKDM4EMAPT
SCHEMBL6945088 0.79 CYP1A2 (0.48) MEN1KMT2ACYP1A2CYP2D6MAPT
SCHEMBL6944405 0.77 F2 (0.48) MEN1KMT2AALDH1A1PNPHRH4
SCHEMBL6950878 0.76 RAB9A (0.53) ALDH1A1MMP2GAAMAPT
SCHEMBL7077175 0.76 DHFR (0.59) MAPT
SCHEMBL6948621 0.76 PNP (0.47) PNPCYP1A2CYP2D6GAAKDM4E
SCHEMBL6941907 0.75 ALDH1A1 (0.47) KMT2AALDH1A1CYP2D6
SCHEMBL6949057 0.74 RIPK1 (0.50) MEN1KMT2AALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed