SCHEMBL6944742

SCHEMBL6944742

CC(C)C[C@@H](C(=O)NNc1ccccc1)C(CC=Cc1cccnc1)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
ADAM17 P78536 4/20 0.40
RAB9A P51151 2/20 0.38
GAA P10253 4/20 0.38
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TBXAS1 P24557 1/20 0.36
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
HTT P42858 1/20 0.35
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942710 0.91 ADAM17 (0.46) ADAM17GAAMMP1MMP2MMP3
SCHEMBL6982398 0.88 CHRNB2 (0.45) CHRNB2CHRNA4ADAM17RAB9AMMP1
SCHEMBL6944086 0.82 ADAM17 (0.42) ADAM17GAAMMP1MMP2MMP3
SCHEMBL6941589 0.82 ADAM17 (0.49) CHRNB2CHRNA4ADAM17RAB9AGAA
SCHEMBL6947136 0.80 ADAM17 (0.44) ADAM17RAB9AGAAMMP1MMP2
SCHEMBL6942460 0.80 ADAM17 (0.46) ADAM17MMP1MMP2MMP3MMP7
SCHEMBL6220493 0.78 ADAM17 (0.48) ADAM17MAPTMAPK1KMT2AATM
SCHEMBL6220502 0.78 ADAM17 (0.48) ADAM17MAPTMAPK1KMT2AATM
SCHEMBL6984686 0.78 ADAM17 (0.48) ADAM17MAPTMAPK1KMT2AATM
SCHEMBL6220496 0.78 ADAM17 (0.48) ADAM17MAPTMAPK1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed