SCHEMBL6960939

SCHEMBL6960939

COc1ccc(Cn2c(COCc3ccccc3)nc(C(C)C)c2Sc2cc(Cl)cc(Cl)c2)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.35
MAPT P10636 2/20 0.35
CSF1R P07333 3/20 0.35
P2RX3 P56373 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NTRK1 P04629 2/20 0.34
NTRK2 Q16620 2/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
TRPV6 Q9H1D0 1/20 0.33
KDR P35968 2/20 0.33
EPHB4 P54760 1/20 0.33
TEK Q02763 1/20 0.33
KMT2A Q03164 1/20 0.32
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
VCP P55072 1/20 0.32
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14439828 0.89 TDP1 (0.40) TP53MAPTTDP1KMT2AVCP
SCHEMBL14439857 0.89 DHODH (0.39) TP53MAPTTDP1
SCHEMBL6957630 0.89 DHODH (0.39) TP53MAPTTDP1
SCHEMBL14002295 0.87 P2RX3 (0.34) CSF1RP2RX3KDREPHB4TEK
SCHEMBL6966431 0.85 TP53 (0.37) TP53MAPTTDP1VCP
SCHEMBL5853114 0.85 TDP1 (0.37) TP53MAPTTDP1TLR7VCP
SCHEMBL6973428 0.84 GABRA1 (0.36) TP53MAPTTDP1KMT2A
SCHEMBL6974703 0.84 TDP1 (0.41) TP53MAPTTDP1KMT2AVCP
SCHEMBL6972460 0.83 P2RX3 (0.36) TP53MAPTP2RX3TDP1VCP
SCHEMBL6966496 0.83 VCP (0.37) TP53MAPTTDP1VCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed