SCHEMBL6964071

SCHEMBL6964071

CC(C)c1nc(CO)n(Cc2ccccc2[N+](=O)[O-])c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TSHR P16473 1/20 0.35
CCR5 P51681 1/20 0.35
CASP1 P29466 1/20 0.35
CASP4 P49662 1/20 0.35
CASP5 P51878 1/20 0.35
CA12 O43570 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
AGTR1 P30556 1/20 0.34
AGTR2 P50052 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
USP7 Q93009 1/20 0.34
ENPP2 Q13822 1/20 0.33
ACHE P22303 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972629 0.93 AGTR1 (0.37) ALDH1A1TSHRCCR5CASP1CASP4
SCHEMBL6960943 0.86 AGTR1 (0.35) ALDH1A1CCR5KDM4ELMNATDP1
SCHEMBL6962626 0.84 AGTR1 (0.34) ALDH1A1CCR5CASP1CASP4CASP5
SCHEMBL6961345 0.84 L3MBTL1 (0.39) ALDH1A1KDM4EMEN1POLBKMT2A
SCHEMBL6960543 0.84 GCGR (0.33) ALDH1A1TSHRKDM4ELMNATDP1
SCHEMBL6970372 0.83 CCR2 (0.43) ALDH1A1KDM4ELMNATDP1MEN1
SCHEMBL6966848 0.82 TDP1 (0.42) ALDH1A1KDM4ETDP1MEN1POLB
Hydrochloric Acid SCHEMBL6970533 0.82 CYP2C19 (0.41) ALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL6969480 0.82 CCR2 (0.43) ALDH1A1KDM4ELMNATDP1MEN1
SCHEMBL6968197 0.80 P2RX3 (0.36) ALDH1A1KDM4ETDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed