SCHEMBL6972629

SCHEMBL6972629

CC(C)c1nc(CCO)n(Cc2ccccc2[N+](=O)[O-])c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.37
AGTR2 P50052 1/20 0.37
CCR5 P51681 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
CASP4 P49662 1/20 0.34
CASP5 P51878 1/20 0.34
DHODH Q02127 1/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
USP7 Q93009 1/20 0.33
DPP4 P27487 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964071 0.93 ALDH1A1 (0.35) AGTR1AGTR2CCR5ALDH1A1TSHR
SCHEMBL6960943 0.88 AGTR1 (0.35) AGTR1AGTR2CCR5ALDH1A1KDM4E
SCHEMBL6962626 0.86 AGTR1 (0.34) AGTR1AGTR2CCR5ALDH1A1CASP1
SCHEMBL6969108 0.84 TSHR (0.38) TSHRKDM4EMEN1KMT2A
SCHEMBL6969846 0.84 KDM4E (0.33) ALDH1A1KDM4ELMNATDP1
SCHEMBL6962951 0.83 CCR2 (0.42) ALDH1A1KDM4ELMNATDP1MEN1
SCHEMBL6970972 0.81 HRH1 (0.31)
SCHEMBL6967398 0.79 HSP90B1 (0.33) KMT2A
SCHEMBL6968855 0.79 ALDH1A1 (0.36) ALDH1A1KDM4ELMNATDP1
SCHEMBL6972122 0.79 PIN1 (0.33) CCR5ALDH1A1CASP1CASP4CASP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP claimed
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed