SCHEMBL6975865

SCHEMBL6975865

Cc1ccc2nc(C(=O)CC(=O)C(F)(F)F)sc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.51
ACP1 P24666 1/20 0.49
DYRK1A Q13627 1/20 0.49
NPC1 O15118 8/20 0.47
RAB9A P51151 8/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
ALDH1A1 P00352 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAOB P27338 3/20 0.46
LMNA P02545 3/20 0.46
GAA P10253 1/20 0.46
PTPN1 P18031 1/20 0.45
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
MAP3K5 Q99683 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975976 0.90 ACP1 (0.47) TP53ACP1DYRK1ANPC1RAB9A
SCHEMBL6982879 0.85 PDPK1 (0.49) DYRK1ANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6983733 0.84 DYRK1A (0.48) DYRK1ANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6979367 0.84 MAPT (0.57) TP53DYRK1ANPC1RAB9ASMN1; SMN2
SCHEMBL6984031 0.83 ACP1 (0.50) TP53ACP1DYRK1ANPC1RAB9A
SCHEMBL6979211 0.81 RAB9A (0.58) TP53NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL6969298 0.81 STING1 (0.39) MAOBGAA
SCHEMBL6981786 0.77 DYRK1A (0.49) DYRK1ANPC1RAB9ASMN1; SMN2MAOB
SCHEMBL6980043 0.75 DYRK1A (0.60) TP53ACP1DYRK1ANPC1RAB9A
SCHEMBL2210476 0.75 DYRK1A (0.56) TP53ACP1DYRK1ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed