SCHEMBL6971808

SCHEMBL6971808

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)CCCC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.40
CACNA1F O60840 2/20 0.40
DRD4 P21917 2/20 0.40
DRD5 P21918 2/20 0.40
HRH2 P25021 2/20 0.40
ADRA1D P25100 2/20 0.40
HTR2A P28223 2/20 0.40
ADRA1A P35348 2/20 0.40
HRH1 P35367 2/20 0.40
ADRA1B P35368 2/20 0.40
OPRM1 P35372 2/20 0.40
DRD3 P35462 2/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40
HTR6 P50406 2/20 0.40
CACNA1D Q01668 2/20 0.40
SLC6A3 Q01959 2/20 0.40
CACNA1S Q13698 2/20 0.40
CACNA1C Q13936 2/20 0.40
DRD1 P21728 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983244 0.95 CACNA1B (0.35) HTR7CACNA1FDRD4DRD5HRH2
SCHEMBL6980780 0.89 CACNA2D1 (0.43) CACNA1CCACNA1G
SCHEMBL6974100 0.88 NPC1 (0.48) HTR7CACNA1FDRD4DRD5HRH2
SCHEMBL6977655 0.85 TSHR (0.47) NPC1RAB9ASIGMAR1
Hydrochloric Acid SCHEMBL6982801 0.85 SIGMAR1 (0.41) HTR7DRD4DRD5HRH2HTR2A
SCHEMBL6975992 0.84 TSHR (0.44)
Hydrochloric Acid SCHEMBL6978285 0.84 SIGMAR1 (0.42) SIGMAR1
Hydrochloric Acid SCHEMBL6984860 0.83 OPRL1 (0.37) OPRM1OPRK1SIGMAR1
SCHEMBL6976114 0.82 USP2 (0.32) ADRA1DHRH1OPRM1DRD3SLC6A3
SCHEMBL9698183 0.79 OPRM1 (0.38) HTR7ADRA1DHTR2AADRA1AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed