SCHEMBL6983244

SCHEMBL6983244

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)CCC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 4/20 0.35
CACNA1C Q13936 3/20 0.35
OPRK1 P41145 2/20 0.35
CACNA1F O60840 1/20 0.35
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD5 P21918 1/20 0.35
HRH2 P25021 1/20 0.35
ADRA1D P25100 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
ADRA1A P35348 1/20 0.35
HRH1 P35367 1/20 0.35
ADRA1B P35368 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
OPRD1 P41143 1/20 0.35
HTR5A P47898 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971808 0.95 HTR7 (0.40) CACNA1COPRK1CACNA1FDRD1DRD4
SCHEMBL6980780 0.91 CACNA2D1 (0.43) CACNA1BCACNA1CCACNA2D1CACNB1
SCHEMBL6977655 0.87 TSHR (0.47)
SCHEMBL6975992 0.86 TSHR (0.44)
SCHEMBL6974100 0.85 NPC1 (0.48) CACNA1COPRK1CACNA1FDRD1DRD4
Hydrochloric Acid SCHEMBL6984860 0.85 OPRL1 (0.37) OPRK1OPRM1
SCHEMBL6976114 0.83 USP2 (0.32) ADRA1DHTR2CHRH1OPRM1DRD3
Hydrochloric Acid SCHEMBL6982801 0.83 SIGMAR1 (0.41) OPRK1DRD1DRD4DRD5HRH2
Hydrochloric Acid SCHEMBL6978285 0.82 SIGMAR1 (0.42) CACNA1B
SCHEMBL9698183 0.81 OPRM1 (0.38) OPRK1DRD1ADRA1DHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed