SCHEMBL6977655

SCHEMBL6977655

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)CCc3ccccc3)CC1)O2

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.45
FKBP1A P62942 1/20 0.43
NPC1 O15118 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
POLB P06746 2/20 0.43
SIGMAR1 Q99720 3/20 0.42
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ME2 P23368 1/20 0.40
ME1 P48163 1/20 0.40
ME3 Q16798 1/20 0.40
MAPT P10636 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
GFER P55789 1/20 0.39
AR P10275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974100 0.94 NPC1 (0.48) TSHRL3MBTL1FKBP1ANPC1POLB
SCHEMBL6971808 0.85 HTR7 (0.40) NPC1SIGMAR1RAB9A
SCHEMBL6981065 0.85 SIGMAR1 (0.41) SIGMAR1MAPTALDH1A1SMN1; SMN2KMT2A
SCHEMBL6980780 0.85 CACNA2D1 (0.43) TSHRTDP1
SCHEMBL8578227 0.83 SIGMAR1 (0.46) POLBSIGMAR1KMT2AMEN1
SCHEMBL6985365 0.83 LMNA (0.42) NPC1POLBSIGMAR1RAB9AALDH1A1
Hydrochloric Acid SCHEMBL6984004 0.82 SIGMAR1 (0.45) POLBSIGMAR1ALDH1A1SMN1; SMN2KMT2A
Hydrochloric Acid SCHEMBL6979044 0.82 LMNA (0.41) TSHRNPC1POLBSIGMAR1RAB9A
Hydrochloric Acid SCHEMBL6982193 0.82 SIGMAR1 (0.45) SIGMAR1
SCHEMBL6976496 0.80 CARM1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed