SCHEMBL6975992

SCHEMBL6975992

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(C(=O)C(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 4/20 0.41
LMNA P02545 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HTT P42858 2/20 0.39
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2D6 P10635 1/20 0.38
GAA P10253 2/20 0.37
TP53 P04637 1/20 0.37
P2RX7 Q99572 1/20 0.36
ADRB2 P07550 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980780 0.88 CACNA2D1 (0.43) TSHRGAA
SCHEMBL6983244 0.86 CACNA1B (0.35)
SCHEMBL6971808 0.84 HTR7 (0.40)
SCHEMBL6976114 0.84 USP2 (0.32) TSHRALDH1A1KDM4ELMNANPSR1
SCHEMBL9698183 0.83 OPRM1 (0.38) ALDH1A1LMNANPSR1MEN1KMT2A
Hydrochloric Acid SCHEMBL8713715 0.82 MEN1 (0.38) ALDH1A1LMNANPSR1MEN1KMT2A
Hydrochloric Acid SCHEMBL6984860 0.81 OPRL1 (0.37) CYP2D6
SCHEMBL6981792 0.80 POLB (0.47) TSHRALDH1A1KDM4ELMNAMEN1
SCHEMBL6974100 0.80 NPC1 (0.48) TSHRALDH1A1KDM4ENPSR1HTT
Hydrochloric Acid SCHEMBL6982801 0.80 SIGMAR1 (0.41) LMNAMEN1KMT2ACYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed