SCHEMBL6974903

SCHEMBL6974903

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccccc4)c32)c(N)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
PKM P14618 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NR3C1 P04150 2/20 0.37
AR P10275 1/20 0.37
CCKBR P32239 1/20 0.37
PTGES2 Q9H7Z7 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
AKR1C3 P42330 2/20 0.35
AKR1C1 Q04828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085529 0.89 MAPT (0.39) TP53LMNAMAPTTHRBPKM
SCHEMBL6983505 0.87 NR3C1 (0.42) TP53LMNAMAPTTHRBPKM
SCHEMBL6985322 0.87 GAA (0.41) TP53LMNAMAPTTHRBPKM
SCHEMBL6974898 0.85 NR3C1 (0.52) TP53LMNAMAPTMEN1KMT2A
SCHEMBL6982953 0.82 CCR10 (0.39) TP53LMNAMAPTPKMMEN1
SCHEMBL6976883 0.81 NR3C1 (0.38) TP53LMNAMAPTTHRBPKM
SCHEMBL6980541 0.80 HSD17B10 (0.48) TP53LMNAMAPTPKMMEN1
SCHEMBL6984039 0.80 TP53 (0.45) TP53LMNAMAPTTHRBPKM
SCHEMBL7411038 0.80 PKM (0.43) TP53LMNAMAPTTHRBPKM
SCHEMBL6977498 0.80 CCKBR (0.44) TP53LMNAMAPTTHRBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed