SCHEMBL6975773

SCHEMBL6975773

Cc1ccc(C2(N3CCOCC3)C=C(C(N)=O)C=CN2)cc1NC(=O)c1cccc(OC2CCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.38
CHEK2 O96017 1/20 0.36
TOP2A P11388 1/20 0.36
OPRK1 P41145 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TBK1 Q9UHD2 1/20 0.34
POLB P06746 2/20 0.34
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973782 0.96 TBK1 (0.36) RAB9ACHEK2TOP2AOPRK1ALDH1A1
SCHEMBL6979960 0.94 CHEK2 (0.41) CHEK2TOP2AKMT2ATBK1
SCHEMBL6972610 0.90 PDE4D (0.41) TOP2AALDH1A1MEN1KMT2ATBK1
SCHEMBL6969085 0.80 CHRM3 (0.37) RAB9AALDH1A1TSHRSMN1; SMN2MEN1
SCHEMBL6975780 0.76 TBK1 (0.43) RAB9ACHEK2OPRK1ALDH1A1TSHR
SCHEMBL6476766 0.76 OPRK1 (0.59) OPRK1ALDH1A1TSHR
SCHEMBL2972096 0.75 OPRK1 (0.58) OPRK1
SCHEMBL7804552 0.74 OPRK1 (0.54) RAB9AOPRK1ALDH1A1TSHRSMN1; SMN2
SCHEMBL6975779 0.73 MAPK14 (0.58)
SCHEMBL6477083 0.72 MAPK14 (0.54) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115707-B1 BENZAMIDE DERIVATIVES AND THER USE AS CYTOKINE INHIBITORS ASTRAZENECA AB (SE) 2003-11-12 EP disclosed