SCHEMBL6975892

SCHEMBL6975892

CC(C)c1nc(CCCO)n(Cc2cnc3ccccc3c2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
FAAH O00519 5/20 0.35
TLR7 Q9NYK1 1/20 0.33
ITGB2 P05107 4/20 0.32
ICAM1 P05362 4/20 0.32
ITGAL P20701 4/20 0.32
TSHR P16473 2/20 0.32
ERCC5 P28715 1/20 0.32
FEN1 P39748 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CNR2 P34972 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967535 0.95 FAAH (0.35) FAAHITGB2ICAM1ITGALERCC5
SCHEMBL6968913 0.91 FAAH (0.36) FAAHITGB2ICAM1ITGALERCC5
SCHEMBL7084086 0.90 TDP1 (0.36) ALDH1A1TDP1FAAHTLR7ITGB2
SCHEMBL7079248 0.87 TDP1 (0.37) ALDH1A1TDP1TLR7
SCHEMBL6972767 0.85 FAAH (0.35) FAAHITGB2ICAM1ITGALERCC5
SCHEMBL6972940 0.84 FAAH (0.35) TDP1FAAHITGB2ICAM1ITGAL
SCHEMBL6974151 0.83 FAAH (0.36) FAAHITGB2ICAM1ITGALERCC5
SCHEMBL7086853 0.83 GRIN1 (0.37) ALDH1A1TDP1TLR7PKM
SCHEMBL6969774 0.82 ENPP2 (0.35) ALDH1A1TDP1TLR7
SCHEMBL6973869 0.82 TLR7 (0.35) ALDH1A1TDP1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed