SCHEMBL6974151

SCHEMBL6974151

CC(C)c1nc(COC(N)=O)n(Cc2cnc3ccccc3c2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 9/20 0.36
ENPP2 Q13822 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
ITGB2 P05107 5/20 0.35
ICAM1 P05362 5/20 0.35
ITGAL P20701 5/20 0.35
ERCC5 P28715 1/20 0.34
FEN1 P39748 1/20 0.34
HCRTR1 O43613 2/20 0.33
HCRTR2 O43614 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972767 0.92 FAAH (0.35) FAAHDPP4DPP8ITGB2ICAM1
SCHEMBL6969844 0.90 FAAH (0.36) FAAHDPP4DPP8ITGB2ICAM1
SCHEMBL6975183 0.88 ENPP2 (0.35) ENPP2
SCHEMBL6968913 0.86 FAAH (0.36) FAAHITGB2ICAM1ITGALERCC5
SCHEMBL6967535 0.85 FAAH (0.35) FAAHENPP2ITGB2ICAM1ITGAL
SCHEMBL6967126 0.84 GRIN1 (0.37) ENPP2
SCHEMBL6973048 0.84 ENPP2 (0.35) ENPP2
SCHEMBL6974519 0.84 ENPP2 (0.35) ENPP2
SCHEMBL7084640 0.83 S1PR3 (0.39) ENPP2
SCHEMBL6975892 0.83 ALDH1A1 (0.36) FAAHITGB2ICAM1ITGALERCC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed