SCHEMBL6987767

SCHEMBL6987767

CCOC(=O)CN(c1cccc2c1N(C(=O)CCc1ccc(C#N)cc1)CCC2)S(=O)(=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
PTGER1 P34995 2/20 0.39
LMNA P02545 2/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HCRTR2 O43614 1/20 0.37
KDM1A O60341 1/20 0.36
ALOX5 P09917 1/20 0.36
TEAD1 P28347 1/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982234 0.87 TP53 (0.41) TP53LMNAUSP2ALDH1A1L3MBTL1
SCHEMBL6986000 0.87 NR3C1 (0.36) LMNAALDH1A1L3MBTL1GAANR3C1
SCHEMBL6982667 0.86 NR3C1 (0.41) TP53KEAP1NFE2L2LMNAUSP2
SCHEMBL7407619 0.86 MAPT (0.34) TP53PTGER1ALDH1A1HCRTR2KDM1A
SCHEMBL6977636 0.86 ALDH1A1 (0.42) TP53LMNAUSP2ALDH1A1GAA
SCHEMBL6982692 0.86 L3MBTL1 (0.38) LMNAALDH1A1L3MBTL1KDM1ANR3C1
SCHEMBL6987763 0.86 NR3C1 (0.47) LMNAUSP2ALDH1A1HCRTR2KDM1A
SCHEMBL6985399 0.85 NOTUM (0.36) LMNAUSP2ALDH1A1L3MBTL1GAA
SCHEMBL6985613 0.84 CCR5 (0.37) LMNAUSP2ALDH1A1L3MBTL1HSD17B10
SCHEMBL6979151 0.83 USP14 (0.35) USP2ALDH1A1L3MBTL1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed