SCHEMBL6983751

SCHEMBL6983751

N#Cc1ccc(CCC(=O)N2CCCc3cccc(S(=O)(=O)c4ccccc4)c32)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.40
AR P10275 1/20 0.40
GAA P10253 1/20 0.39
NPC1 O15118 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 3/20 0.38
NAAA Q02083 1/20 0.38
FPR1 P21462 2/20 0.37
FPR2 P25090 2/20 0.37
MAPK1 P28482 2/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986981 0.86 MCL1 (0.40) NR3C1ARGAAALDH1A1MEN1
SCHEMBL6985295 0.85 MAPT (0.45) ALDH1A1MEN1KMT2AMAPTFPR1
SCHEMBL6985322 0.84 GAA (0.41) NR3C1ARGAANPC1ALDH1A1
SCHEMBL6977636 0.84 ALDH1A1 (0.42) NR3C1ARGAANPC1ALDH1A1
SCHEMBL6982667 0.82 NR3C1 (0.41) NR3C1ARGAAALDH1A1TSHR
SCHEMBL6983746 0.82 NR3C1 (0.47) NR3C1GAATDP1ALDH1A1TSHR
SCHEMBL6979727 0.81 TSHR (0.40) NPC1ALDH1A1TSHRMEN1USP2
SCHEMBL6977399 0.81 PTGER4 (0.42) NR3C1ARGAANPC1TDP1
SCHEMBL6985566 0.81 PARP14 (0.40) NR3C1ARNPC1TDP1ALDH1A1
SCHEMBL6986002 0.80 RXRA (0.45) ARNPC1TDP1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed