SCHEMBL6981065

SCHEMBL6981065

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCN(CCc3ccccc3)CC1)O2

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.41
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SLC6A3 Q01959 1/20 0.39
DRD2 P14416 2/20 0.39
HTR1A P08908 1/20 0.39
ACHE P22303 1/20 0.38
OPRM1 P35372 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KCNH2 Q12809 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8578227 0.94 SIGMAR1 (0.46) SIGMAR1MEN1KMT2A
Hydrochloric Acid SCHEMBL6984004 0.93 SIGMAR1 (0.45) SIGMAR1ALDH1A1MEN1KMT2ANPSR1
Hydrochloric Acid SCHEMBL6982193 0.92 SIGMAR1 (0.45) SIGMAR1
SCHEMBL6985365 0.89 LMNA (0.42) SIGMAR1ALDH1A1ACHESMN1; SMN2
Hydrochloric Acid SCHEMBL6979044 0.88 LMNA (0.41) SIGMAR1ALDH1A1MEN1KMT2AMAPT
SCHEMBL6976496 0.85 CARM1 (0.42) ACHEKCNH2
SCHEMBL6977655 0.85 TSHR (0.47) SIGMAR1ALDH1A1MEN1KMT2AMAPT
SCHEMBL6983488 0.84 DRD2 (0.41) SIGMAR1ALDH1A1MEN1KMT2AMAPT
SCHEMBL6981074 0.84 HRH3 (0.40) SIGMAR1ACHE
SCHEMBL6974100 0.83 NPC1 (0.48) SIGMAR1ALDH1A1MAPTNPSR1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed