SCHEMBL6979916

SCHEMBL6979916

Nc1nc(Cc2ccc(OCc3ccccc3)cc2)cc(C2CCN(C(=O)c3ccc4c(c3)OCO4)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
TSHR P16473 3/20 0.43
YAP1 P46937 1/20 0.43
EDNRB P24530 2/20 0.43
EDNRA P25101 2/20 0.43
MAOB P27338 1/20 0.42
GFER P55789 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PRMT5 O14744 2/20 0.42
SLC6A7 Q99884 1/20 0.42
KDM4E B2RXH2 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
MCHR1 Q99705 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HPGD P15428 1/20 0.40
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7123772 0.88 SMN1; SMN2 (0.51) ALDH1A1TSHRHSD17B10KMT2AMCHR1
SCHEMBL6980741 0.88 HPGD (0.47) ALDH1A1TSHRGFERHSD17B10KMT2A
SCHEMBL6980066 0.85 ALDH1A1 (0.48) ALDH1A1TSHRHSD17B10KMT2AMEN1
SCHEMBL6972446 0.82 HSD17B10 (0.48) ALDH1A1YAP1HSD17B10LMNASMN1; SMN2
SCHEMBL6976878 0.78 HSD11B1 (0.51) ALDH1A1KMT2AMEN1LMNAHPGD
SCHEMBL6973351 0.76 DRD2 (0.52) ALDH1A1KMT2AMEN1LMNA
SCHEMBL6976438 0.74 NPC1 (0.45) KMT2ALMNA
SCHEMBL6975639 0.72 MAP3K12 (0.49) KMT2AMEN1LMNA
SCHEMBL8392370 0.70 MAOB (0.41) ALDH1A1EDNRBEDNRAMAOBLMNA
SCHEMBL6981142 0.70 GLA (0.55) TSHRKMT2AMEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892795-B1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMA (JP) 2003-01-08 EP disclosed
EP-0892795-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1999-01-27 EP disclosed
WO-1997038992-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-23 WO disclosed