SCHEMBL6981485

SCHEMBL6981485

O=C(O)C1(c2cccs2)OCC2(CO1)c1ccccc1-c1ccccc12

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 3/20 0.37
HCAR2 Q8TDS4 1/20 0.34
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
LMNA P02545 2/20 0.33
PDK2 Q15119 2/20 0.33
OPRM1 P35372 2/20 0.32
OPRL1 P41146 2/20 0.32
APEX1 P27695 1/20 0.32
MAPT P10636 2/20 0.32
KMT2A Q03164 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
ITGA4 P13612 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983335 0.82 HSD17B10 (0.38) ALDH1A1LMNAMAPTKMT2A
SCHEMBL7831174 0.81 HSD11B1 (0.36) ALDH1A1HTTLMNAOPRM1MAPT
SCHEMBL6982681 0.80 THRB (0.44) THRBTDP1ALDH1A1PDK2APEX1
SCHEMBL6971210 0.74 CYP1A2 (0.41) THRBTDP1TP53HTTLMNA
SCHEMBL6982212 0.72 THRB (0.46) THRBTDP1ALDH1A1LMNAPDK2
SCHEMBL6971971 0.71 NPC1 (0.44) ALDH1A1TP53PDK2OPRM1OPRL1
SCHEMBL6633029 0.70 ALDH1A1 (0.42) ALDH1A1HCAR2TP53HTTLMNA
SCHEMBL6968252 0.69 MEN1 (0.42) THRBTDP1ALDH1A1HTTLMNA
SCHEMBL6978402 0.69 OPRM1 (0.41) OPRM1OPRL1OPRD1OPRK1GAA
SCHEMBL6981621 0.67 APEX1 (0.42) THRBTDP1ALDH1A1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098893-B1 CYCLIC COMPOUNDS USEFUL IN THE TREATMENT OF DYSLIPIDEMIA, ATHEROSCLEROSIS AND DIABETES, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PROCESS MERCK PATENT GMBH (DE) 2003-03-26 EP disclosed