SCHEMBL6981764

SCHEMBL6981764

NCc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccc(F)cc4)c32)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.42
GAA P10253 5/20 0.42
SLC16A3 O15427 1/20 0.41
ALDH1A1 P00352 9/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PKM P14618 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPT P10636 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
HTT P42858 1/20 0.39
MGAT2 Q10469 1/20 0.38
DNMT1 P26358 1/20 0.38
CASP6 P55212 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984843 0.92 GAA (0.43) METAP2GAAALDH1A1MEN1KMT2A
SCHEMBL6984822 0.91 SLC16A3 (0.40) METAP2GAASLC16A3ALDH1A1MEN1
SCHEMBL6982764 0.90 FPR1 (0.43) METAP2GAASLC16A3ALDH1A1MEN1
SCHEMBL6982500 0.82 SLC16A3 (0.48) GAASLC16A3
SCHEMBL6982743 0.82 F2 (0.42) METAP2GAA
SCHEMBL6985322 0.81 GAA (0.41) METAP2GAAALDH1A1MEN1KMT2A
SCHEMBL6981763 0.81 BRD4 (0.54) ALDH1A1MEN1KMT2ALMNASMN1; SMN2
SCHEMBL6985749 0.81 ALDH1A1 (0.48) GAAALDH1A1MEN1KMT2ALMNA
SCHEMBL6984759 0.81 LMNA (0.47) GAAALDH1A1MEN1KMT2ALMNA
SCHEMBL7408050 0.81 TP53 (0.40) GAAALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed