SCHEMBL6984787

SCHEMBL6984787

NCc1ccc(CCC(=O)N2CCCc3cccc(NC(=O)c4ccccc4)c32)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.48
POLB P06746 1/20 0.44
RECQL P46063 1/20 0.44
KDM1A O60341 3/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 2/20 0.40
HDAC1 Q13547 2/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985381 0.89 MMP1 (0.45) ATMPOLBRECQLKDM1ARAB9A
SCHEMBL6984843 0.82 GAA (0.43) POLBRAB9AMEN1ALDH1A1KMT2A
SCHEMBL6984783 0.80 RAB9A (0.64) POLBRAB9AALDH1A1MAPTNPC1
SCHEMBL6982500 0.77 SLC16A3 (0.48) POLB
SCHEMBL6986817 0.76 THRB (0.42) ATMPOLBALDH1A1MAPTKMT2A
SCHEMBL6981837 0.76 AVPR2 (0.39) ATMRAB9AMEN1ALDH1A1MAPT
SCHEMBL6981764 0.76 METAP2 (0.42) MEN1ALDH1A1MAPTKMT2AKDM4E
SCHEMBL6982743 0.75 F2 (0.42)
SCHEMBL6977743 0.74 PTGER4 (0.46) POLBRECQLMEN1ALDH1A1MAPT
SCHEMBL6980994 0.74 RXRA (0.43) ATMRAB9AMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed