SCHEMBL6983767

SCHEMBL6983767

CC(C)n1nc(-c2cc(N3CCN(Cc4ccccc4)CC3)nn2-c2ccccc2)ccc1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.41
MGLL Q99685 1/20 0.40
DRD2 P14416 2/20 0.40
CASP1 P29466 1/20 0.39
CASP5 P51878 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 2/20 0.38
KDM4E B2RXH2 1/20 0.38
USP2 O75604 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KHK P50053 1/20 0.38
SMO Q99835 1/20 0.38
DPP4 P27487 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981026 0.89 AGTR2 (0.40) MGLLTSHRALDH1A1MAPTLMNA
SCHEMBL6984622 0.87 AGTR2 (0.39) MGLLCASP1TSHRALDH1A1LMNA
SCHEMBL6986283 0.85 HTR2C (0.42) DRD2KHKAGTR2
SCHEMBL6988437 0.84 ALDH1A1 (0.45) TSHRALDH1A1LMNANPC1RAB9A
SCHEMBL6981802 0.83 ALDH1A1 (0.42) TSHRALDH1A1MAPTNPSR1LMNA
SCHEMBL6986113 0.83 AGTR2 (0.41) MGLLALDH1A1LMNAUSP2HSD17B10
SCHEMBL6986237 0.82 AGTR2 (0.39) ALDH1A1MAPTNPSR1LMNAKDM4E
SCHEMBL6988584 0.82 USP2 (0.43) MGLLTSHRALDH1A1MAPTLMNA
SCHEMBL6983724 0.81 MEN1 (0.39) TSHRMAPTLMNAKDM4EUSP2
SCHEMBL6984642 0.80 HRH3 (0.39) AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313733-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-28 EP disclosed
WO-2002018382-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-03-07 WO disclosed