SCHEMBL6988437

SCHEMBL6988437

CC(C)n1nc(-c2cc(N3CCOCC3)nn2-c2ccccc2)ccc1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PIK3C3 Q8NEB9 1/20 0.42
LMNA P02545 1/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
BRD4 O60885 1/20 0.39
PIK3CB P42338 6/20 0.38
PIK3CD O00329 4/20 0.38
PIK3CA P42336 4/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
PIK3R1 P27986 1/20 0.38
CSNK1A1 P48729 1/20 0.38
PIK3CG P48736 1/20 0.38
PTK2 Q05397 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981026 0.92 AGTR2 (0.40) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL6986283 0.88 HTR2C (0.42)
SCHEMBL6984622 0.88 AGTR2 (0.39) ALDH1A1SMN1; SMN2LMNAKMT2ABRD4
SCHEMBL6986237 0.85 AGTR2 (0.39) ALDH1A1LMNAMEN1KMT2APIK3CB
SCHEMBL6981802 0.85 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL6986113 0.85 AGTR2 (0.41) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL6983767 0.84 DRD4 (0.41) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL6984642 0.84 HRH3 (0.39) BRD4CFTR
SCHEMBL6984282 0.83 HSD17B10 (0.43) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL6988584 0.83 USP2 (0.43) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313733-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-28 EP disclosed
WO-2002018382-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-03-07 WO disclosed