SCHEMBL6986237

SCHEMBL6986237

CC(C)n1nc(-c2cc(N3CCC(O)CC3)nn2-c2ccccc2)ccc1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.39
CFTR P13569 1/20 0.36
PHGDH O43175 1/20 0.35
HSD11B1 P28845 1/20 0.35
HRH3 Q9Y5N1 3/20 0.34
ALDH1A1 P00352 3/20 0.34
GAA P10253 3/20 0.34
MYC P01106 2/20 0.34
WDR5 P61964 2/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
GLA P06280 2/20 0.33
POLB P06746 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33
SLC5A1 P13866 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981026 0.88 AGTR2 (0.40) AGTR2HSD11B1HRH3ALDH1A1KDM4E
SCHEMBL6984642 0.88 HRH3 (0.39) AGTR2CFTRHSD11B1HRH3
SCHEMBL6986283 0.86 HTR2C (0.42) AGTR2
SCHEMBL6984622 0.86 AGTR2 (0.39) AGTR2HRH3ALDH1A1POLBKMT2A
SCHEMBL6988437 0.85 ALDH1A1 (0.45) CFTRALDH1A1GAAMEN1KMT2A
SCHEMBL6986113 0.85 AGTR2 (0.41) AGTR2ALDH1A1GAAMEN1KMT2A
SCHEMBL6988584 0.83 USP2 (0.43) AGTR2HRH3ALDH1A1MEN1POLB
SCHEMBL6981802 0.83 ALDH1A1 (0.42) AGTR2ALDH1A1GAAKDM4EMEN1
SCHEMBL6983767 0.82 DRD4 (0.41) AGTR2ALDH1A1KDM4EMEN1POLB
SCHEMBL6984282 0.81 HSD17B10 (0.43) ALDH1A1GAAMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313733-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-28 EP disclosed
WO-2002018382-A1 PYRAZOLOPYRIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-03-07 WO disclosed