SCHEMBL6989674

SCHEMBL6989674

CC(C)(CNC(=O)CCc1ccccc1)CNc1c(Nc2cccnc2)c(=O)c1=O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ALDH1A1 P00352 4/20 0.43
HTT P42858 1/20 0.42
PAX8 Q06710 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
KCNA5 P22460 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NOTUM Q6P988 1/20 0.40
LMNA P02545 1/20 0.40
NAMPT P43490 1/20 0.39
TBXA2R P21731 1/20 0.39
TBXAS1 P24557 1/20 0.39
BCL6 P41182 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146201 0.90 LMNA (0.44) CYP1A2CYP3A4CYP2C9ALDH1A1MAPKAPK2
SCHEMBL6986925 0.81 MEN1 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6989669 0.78 CYP3A4 (0.45) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6988180 0.78 NAMPT (0.51) ALDH1A1HTTSMN1; SMN2LMNANAMPT
SCHEMBL6981925 0.77 NAMPT (0.50) CYP1A2CYP3A4CYP2C9CYP2C19HTT
SCHEMBL6988688 0.77 ABCC9 (0.41) MAPKAPK2NOTUMLMNANAMPTTBXA2R
SCHEMBL6990458 0.77 CSF1R (0.44) ALDH1A1MAPKAPK2LMNANAMPTTBXA2R
SCHEMBL7092751 0.76 CYP3A4 (0.43) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6987131 0.75 GRM5 (0.44) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL6988714 0.75 SIRT2 (0.43) ALDH1A1MAPKAPK2TBXA2RTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358160-A1 AMINAL DIONES AS POTASSIUM CHANNEL OPENERS Abbott Laboratories (US) 2003-11-05 EP disclosed
WO-2002062761-A1 AMINAL DIONES AS POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2002-08-15 WO disclosed