SCHEMBL7003350

SCHEMBL7003350

COc1ccc(C(c2cccc(C(F)(F)F)c2)c2c(CO)[nH]c3ccccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VDR P11473 4/20 0.47
CNR1 P21554 3/20 0.43
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
ALOX15 P16050 1/20 0.38
ALOX12 P18054 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KIF11 P52732 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003963 0.82 VDR (0.47) VDRCNR1NR3C1PGRNR3C2
SCHEMBL7003917 0.81 KMT2A (0.54) VDRKDM4EALDH1A1MAPTLMNA
SCHEMBL11201464 0.69 KMT2A (0.54) KDM4EALDH1A1MAPTLMNAGAA
SCHEMBL2010410 0.67 IDO1 (0.47) KDM4EALDH1A1MAPTLMNAGAA
SCHEMBL11193839 0.67 ALDH1A1 (0.48) ALDH1A1MAPTLMNAGAAMEN1
Hydrochloric Acid SCHEMBL2013413 0.66 IDO1 (0.49) KDM4EALDH1A1MAPTLMNAGAA
SCHEMBL7377758 0.64 CCNB2 (0.49) VDRKDM4EALDH1A1LMNAGLA
SCHEMBL29443497 0.64 KIF11 (0.46) KDM4EALDH1A1LMNAGLAGAA
SCHEMBL11272541 0.64 FFAR4 (0.48) CNR1KDM4ELMNAGAAMEN1
SCHEMBL11050404 0.64 MAOB (0.47) KDM4EALDH1A1MAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1341761-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2003-09-10 EP disclosed
WO-2002030895-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-η BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-18 WO disclosed