SCHEMBL7003963

SCHEMBL7003963

COc1ccc(C(c2cccc(C(F)(F)F)c2)c2c(C=O)[nH]c3ccccc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
VDR P11473 5/20 0.47
CNR1 P21554 4/20 0.43
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
ABCG2 Q9UNQ0 2/20 0.40
KIF11 P52732 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP19A1 P11511 1/20 0.38
MAOB P27338 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003350 0.82 VDR (0.47) VDRCNR1NR3C1PGRNR3C2
SCHEMBL7003917 0.79 KMT2A (0.54) VDRKDM4EMEN1ALDH1A1MAPT
SCHEMBL11050404 0.71 MAOB (0.47) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL11201464 0.67 KMT2A (0.54) KDM4EMEN1ALDH1A1MAPTKMT2A
SCHEMBL2010410 0.67 IDO1 (0.47) KIF11KDM4EMEN1ALDH1A1MAPT
SCHEMBL11193839 0.67 ALDH1A1 (0.48) MEN1ALDH1A1MAPTKMT2AMAOB
Hydrochloric Acid SCHEMBL2013413 0.66 IDO1 (0.49) KIF11KDM4EMEN1ALDH1A1MAPT
SCHEMBL2592358 0.64 ALDH1A1 (0.50) ABCG2KIF11KDM4EMEN1ALDH1A1
SCHEMBL7372288 0.64 CCNB2 (0.49) VDRKIF11KDM4EMEN1ALDH1A1
SCHEMBL21399702 0.64 NR3C1 (0.62) VDRNR3C1PGRNR3C2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1341761-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-$g(g) BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2003-09-10 EP disclosed
WO-2002030895-A1 SUBSTITUTED INDOLES, PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH INDOLES AND THEIR USE AS PPAR-η BINDING AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2002-04-18 WO disclosed