SCHEMBL7003856

SCHEMBL7003856

CCCCOc1c2cc(=O)c(C(F)(F)F)cc-2cn(CC(C)(C)C)c1C(=O)OCC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
HPGD P15428 3/20 0.31
KDM4E B2RXH2 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
HSD17B10 Q99714 2/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ESR1 P03372 1/20 0.30
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
LMNA P02545 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006171 0.88 ESR1 (0.34) ALDH1A1L3MBTL1THRATHRBHPGD
SCHEMBL7559797 0.84 ALDH1A1 (0.38) ALDH1A1L3MBTL1HPGDKDM4EHSD17B10
SCHEMBL7001088 0.82 NPC1 (0.36) ALDH1A1L3MBTL1HPGDHDAC3HDAC1
SCHEMBL7002285 0.78 MCL1 (0.38) THRATHRBFFAR4
SCHEMBL7006166 0.76 ESR1 (0.38) ALDH1A1L3MBTL1THRATHRBHPGD
SCHEMBL7004077 0.74 SLC6A5 (0.38) ALDH1A1KDM4EMAPT
SCHEMBL7002721 0.74 JMJD6 (0.33) ALDH1A1L3MBTL1HPGDADORA3MAPT
SCHEMBL7005350 0.74 SLC6A5 (0.38) ALDH1A1KDM4ELMNAMAPTSMN1; SMN2
SCHEMBL7555960 0.74 TDP1 (0.38) ALDH1A1HPGDKDM4ENPC1RAB9A
SCHEMBL7007295 0.72 PTPN11 (0.37) ALDH1A1HPGDKDM4EHSD17B10NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A9 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-10-10 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed