SCHEMBL7012844

SCHEMBL7012844

Cn1ncc2c(ccn2Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 3/20 0.47
HDAC3 O15379 2/20 0.47
HDAC2 Q92769 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
VNN1 O95497 3/20 0.41
TP53 P04637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HTT P42858 2/20 0.41
FSCN1 Q16658 1/20 0.39
BPTF Q12830 1/20 0.39
VEGFA P15692 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
FABP6 P51161 1/20 0.38
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016172 0.91 HDAC3 (0.44) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL7016067 0.90 HDAC3 (0.47) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL7017139 0.88 MAPT (0.42) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL7012328 0.87 ALDH1A1 (0.43) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL7010653 0.82 PKM (0.45) SMN1; SMN2LMNAVNN1TP53TDP1
SCHEMBL7019117 0.81 LMNA (0.43) SMN1; SMN2LMNAVNN1HTTKMT2A
SCHEMBL7014669 0.79 HDAC1 (0.42) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL7021991 0.77 HDAC1 (0.42) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL7017977 0.76 TRPA1 (0.50) HDAC6SMN1; SMN2LMNAVNN1HTT
SCHEMBL7011568 0.76 HPGD (0.44) SMN1; SMN2LMNATP53TDP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed