SCHEMBL7015995

SCHEMBL7015995

CCn1cnc2c(c(C)cn2Cc2ccc(C(=O)c3ccccc3CN3CCN(c4ccccc4)CC3)cc2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
HSD17B10 Q99714 2/20 0.40
ADORA1 P30542 1/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HTR7 P34969 2/20 0.37
HTR1A P08908 1/20 0.37
KMT2A Q03164 2/20 0.36
HSD17B13 Q7Z5P4 1/20 0.36
CSF1R P07333 1/20 0.36
HTR6 P50406 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015205 0.80 L3MBTL1 (0.57) MAPTSMN1; SMN2HSD17B10ALDH1A1HTR7
SCHEMBL7017298 0.76 TP53 (0.46) MAPTSMN1; SMN2ALDH1A1KMT2ALMNA
SCHEMBL7021271 0.76 CYP19A1 (0.41) MAPTSMN1; SMN2KMT2AHSD17B13LMNA
SCHEMBL7016056 0.75 THRB (0.47) MAPTSMN1; SMN2ALDH1A1KMT2AHSD17B13
Morpholine SCHEMBL7015362 0.74 NPSR1 (0.36) MAPTSMN1; SMN2ALDH1A1KMT2AHPGD
SCHEMBL7019393 0.74 HTT (0.42) MAPTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL7008880 0.73 TP53 (0.37) MAPTSMN1; SMN2ALDH1A1KMT2AL3MBTL1
Hydrochloric Acid SCHEMBL7015357 0.70 ALDH1A1 (0.36) SMN1; SMN2ALDH1A1KMT2AL3MBTL1LMNA
SCHEMBL7020188 0.68 LMNA (0.46) MAPTSMN1; SMN2HSD17B10ALDH1A1KMT2A
SCHEMBL7015987 0.66 TP53 (0.47) MAPTSMN1; SMN2HSD17B10ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed