SCHEMBL7017128

SCHEMBL7017128

O=C(NCCCCC(=O)N1CCC2OCC(=O)C21)c1ccc(OC(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.44
DPP4 P27487 10/20 0.42
CTSS P25774 4/20 0.42
CTSV O60911 3/20 0.42
CTSL P07711 3/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC3 O15379 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015308 0.85 CTSK (0.46) CTSKCTSSCTSVCTSLKMT2A
SCHEMBL7020985 0.85 CTSK (0.46) CTSKDPP4CTSSCTSVCTSL
SCHEMBL7024341 0.83 NAMPT (0.48) CTSKDPP4CTSSCTSVCTSL
SCHEMBL7016550 0.80 CTSK (0.41) CTSKDPP4CTSSCTSVCTSL
SCHEMBL7019711 0.79 LMNA (0.52) CTSKDPP4CTSSCTSVCTSL
SCHEMBL7021109 0.78 CTSK (0.41) CTSKDPP4CTSSCTSVCTSL
SCHEMBL4451968 0.77 CTSS (0.69) CTSKCTSSCTSVCTSLKMT2A
SCHEMBL4456121 0.77 CTSK (0.74) CTSKCTSSCTSVCTSL
SCHEMBL7016446 0.77 HDAC1 (0.48) CTSKDPP4CTSSCTSVCTSL
SCHEMBL4452934 0.76 CTSK (0.60) CTSKCTSSCTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362052-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-19 EP disclosed
WO-2002057270-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed