SCHEMBL7017131

SCHEMBL7017131

COc1ccc(C(=O)c2ccc(Cn3c(C)c(C)c4c(=O)n(C)ncc43)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.44
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
PDE1B Q01064 8/20 0.43
PDE1A P54750 7/20 0.43
PDE1C Q14123 7/20 0.43
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
NPBWR1 P48145 2/20 0.41
VNN1 O95497 2/20 0.41
MCHR1 Q99705 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HDAC11 Q96DB2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020546 0.88 MAPT (0.41) TP53MAPTHDAC1HDAC8HDAC6
SCHEMBL7015600 0.87 MAPT (0.43) TP53MAPTMEN1KMT2A
SCHEMBL7019092 0.80 MAPT (0.41) TP53MAPTHDAC1HDAC8HDAC6
SCHEMBL7019042 0.72 KAT2B (0.46) TP53MAPTHDAC1HDAC8HDAC6
SCHEMBL7010725 0.70 NPC1 (0.42) MAPTHDAC1HDAC8HDAC6NPBWR1
SCHEMBL14971734 0.67 HPGD (0.54) CYP19A1TP53MAPTGLAGAA
SCHEMBL7010653 0.65 PKM (0.45) TP53MAPTNPBWR1VNN1
SCHEMBL28232519 0.64 RAB9A (0.63) CYP19A1MAPTGAAVNN1MEN1
SCHEMBL24687649 0.63 NPBWR1 (0.75) NPBWR1MCHR1
SCHEMBL19458501 0.63 PDE1B (0.56) MAPTPDE1BPDE1APDE1CNPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed