SCHEMBL7010725

SCHEMBL7010725

Cn1ncc2c(c(Cl)c(Cl)n2Cc2ccc(C(=O)c3ccc(C(F)(F)F)cc3)cc2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
NPBWR1 P48145 1/20 0.39
CCR9 P51686 1/20 0.39
SRD5A2 P31213 2/20 0.39
P2RX3 P56373 1/20 0.38
VNN1 O95497 2/20 0.38
PDE2A O00408 2/20 0.37
PKM P14618 1/20 0.36
PKLR P30613 1/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC8 Q9BY41 3/20 0.36
HDAC6 Q9UBN7 3/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019042 0.89 KAT2B (0.46) NPC1ALDH1A1LMNAMAPTHTT
SCHEMBL7013283 0.88 HTT (0.40) ALDH1A1LMNAMAPTHTTVNN1
SCHEMBL7018851 0.86 PPARG (0.41) NPC1ALDH1A1LMNAMAPTHTT
SCHEMBL7015497 0.80 MAPT (0.42) ALDH1A1LMNAMAPTRAB9ASRD5A2
SCHEMBL7018161 0.80 CCR2 (0.39) NPC1ALDH1A1LMNAMAPTHTT
SCHEMBL7012328 0.77 ALDH1A1 (0.43) NPC1ALDH1A1LMNAMAPTHTT
SCHEMBL7020546 0.74 MAPT (0.41) ALDH1A1LMNAMAPTHTTHDAC1
SCHEMBL7015600 0.74 MAPT (0.43) LMNAMAPT
SCHEMBL7017131 0.70 CYP19A1 (0.44) NPC1MAPTRAB9ANPBWR1VNN1
SCHEMBL7008568 0.68 PKM (0.41) ALDH1A1LMNAMAPTHTTNPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed