SCHEMBL7019042

SCHEMBL7019042

Cn1ncc2c(c(Cl)c(Cl)n2Cc2ccc(C(=O)c3ccc(F)cc3)cc2)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 2/20 0.46
BRD4 O60885 1/20 0.46
HTT P42858 3/20 0.43
NPSR1 Q6W5P4 3/20 0.43
RAB9A P51151 2/20 0.43
PKM P14618 2/20 0.43
MITF O75030 1/20 0.43
BPTF Q12830 1/20 0.40
MAPT P10636 3/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
JAK2 O60674 1/20 0.39
S1PR2 O95136 1/20 0.39
LMNA P02545 1/20 0.39
XBP1 P17861 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
VNN1 O95497 1/20 0.38
POLB P06746 3/20 0.38
TP53 P04637 2/20 0.38
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013283 0.91 HTT (0.40) BRD4HTTNPSR1MITFBPTF
SCHEMBL7010725 0.89 NPC1 (0.42) HTTRAB9APKMMAPTALDH1A1
SCHEMBL7015600 0.85 MAPT (0.43) KAT2BBRD4MAPTLMNAPOLB
SCHEMBL7015497 0.83 MAPT (0.42) RAB9AMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL7018161 0.83 CCR2 (0.39) BRD4HTTNPSR1RAB9ABPTF
SCHEMBL7020546 0.77 MAPT (0.41) HTTMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL7016067 0.76 HDAC3 (0.47) KAT2BBRD4HTTNPSR1RAB9A
SCHEMBL7018851 0.74 PPARG (0.41) HTTRAB9APKMMAPTALDH1A1
SCHEMBL7017131 0.72 CYP19A1 (0.44) RAB9AMAPTNPC1VNN1TP53
SCHEMBL7008568 0.70 PKM (0.41) HTTPKMMITFMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed