SCHEMBL7013283

SCHEMBL7013283

Cn1ncc2c(c(Cl)c(Cl)n2Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 3/20 0.39
ALDH1A1 P00352 3/20 0.39
TP53 P04637 3/20 0.39
MITF O75030 1/20 0.39
S1PR4 O95977 1/20 0.39
S1PR1 P21453 1/20 0.39
VNN1 O95497 2/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
DRD2 P14416 1/20 0.37
TBXA2R P21731 1/20 0.37
POLB P06746 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
BPTF Q12830 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019042 0.91 KAT2B (0.46) HTTSMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL7018161 0.91 CCR2 (0.39) HTTSMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL7015497 0.89 MAPT (0.42) SMN1; SMN2LMNAMAPTALDH1A1TP53
SCHEMBL7010725 0.88 NPC1 (0.42) HTTLMNAMAPTALDH1A1VNN1
SCHEMBL7020546 0.85 MAPT (0.41) HTTSMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL7008568 0.79 PKM (0.41) HTTSMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL7010653 0.77 PKM (0.45) HTTSMN1; SMN2LMNAMAPTALDH1A1
SCHEMBL7012844 0.76 HDAC1 (0.47) HTTSMN1; SMN2LMNAALDH1A1TP53
SCHEMBL7015600 0.76 MAPT (0.43) LMNAMAPTTP53POLBMEN1
SCHEMBL7019092 0.75 MAPT (0.41) HTTSMN1; SMN2MAPTTP53HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed