SCHEMBL7038205

SCHEMBL7038205

N#Cc1c(F)c(C(=O)O)cc(F)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
NOTUM Q6P988 3/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
DAO P14920 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.34
CYP3A4 P08684 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
MAP2K1 Q02750 1/20 0.33
GPR35 Q9HC97 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ASPH Q12797 1/20 0.33
KDM8 Q8N371 1/20 0.33
KDM4A O75164 1/20 0.32
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
STING1 Q86WV6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5361238 0.88 KEAP1 (0.44) KEAP1NFE2L2NOTUMTAS1R3TAS1R1
Hydrochloric Acid SCHEMBL9475356 0.86 KEAP1 (0.43) KEAP1NFE2L2NOTUMTAS1R3TAS1R1
SCHEMBL3552234 0.84 KEAP1 (0.39) KEAP1NFE2L2NOTUMTRPV4MAP2K1
SCHEMBL22972614 0.77 KEAP1 (0.52) KEAP1NFE2L2NOTUMDAOCYP3A4
SCHEMBL5360639 0.77 ALDH1A1 (0.37) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
SCHEMBL5704378 0.76 TAS1R3 (0.35) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
SCHEMBL7038698 0.76 CASP1 (0.39) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
SCHEMBL18149189 0.74 NOTUM (0.43) NOTUMTAS1R3TAS1R1TAS1R2MRGPRX4
SCHEMBL29376622 0.74 KEAP1 (0.52) KEAP1NFE2L2NOTUMDAOCYP3A4
SCHEMBL2434231 0.74 KEAP1 (0.52) KEAP1NFE2L2NOTUMDAOCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001929-B1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID BAYER AG (DE) 2003-03-26 EP disclosed
US-6462218-B1 BY HYDROLYTIC CLEAVAGE CARRIED OUT IN THE PRESENCE OF ACIDS AND WATER OF ITS AMIDE, ESTER OR CYANO DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed