SCHEMBL7038698

SCHEMBL7038698

N#Cc1c(Cl)c(F)cc(C(N)=O)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 4/20 0.39
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
DGAT1 O75907 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KHK P50053 1/20 0.34
TRPV4 Q9HBA0 1/20 0.33
ADRA1D P25100 2/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5360639 0.84 ALDH1A1 (0.37) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
SCHEMBL5361238 0.84 KEAP1 (0.44) CASP1KEAP1NFE2L2TAS1R3TAS1R1
SCHEMBL5704378 0.83 TAS1R3 (0.35) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
Hydrochloric Acid SCHEMBL9475356 0.83 KEAP1 (0.43) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
SCHEMBL7038205 0.76 KEAP1 (0.43) KEAP1NFE2L2TAS1R3TAS1R1TAS1R2
SCHEMBL10617319 0.76 KEAP1 (0.41) CASP1KEAP1NFE2L2DGAT1MEN1
SCHEMBL7044003 0.75 DGAT1 (0.38) CASP1DGAT1TAS1R3TAS1R1TAS1R2
SCHEMBL9899980 0.74 KEAP1 (0.40) CASP1KEAP1NFE2L2DGAT1MEN1
SCHEMBL5704384 0.72 ALDH1A1 (0.41) MEN1ALDH1A1KMT2ATP53CYP3A4
SCHEMBL9790158 0.71 ALDH1A1 (0.44) TAS1R3TAS1R1TAS1R2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001929-B1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID BAYER AG (DE) 2003-03-26 EP disclosed
US-6462218-B1 BY HYDROLYTIC CLEAVAGE CARRIED OUT IN THE PRESENCE OF ACIDS AND WATER OF ITS AMIDE, ESTER OR CYANO DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed
EP-1001929-A1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID Bayer Aktiengesellschaft (DE) 2000-05-24 EP disclosed
WO-1999006360-A1 METHOD FOR PREPARING 3-CYANO-2,4-DIHALOGEN-5-FLUOR-BENZOIC ACID BAYER AKTIENGESELLSCHAFT (DE) 1999-02-11 WO disclosed