SCHEMBL7058052

SCHEMBL7058052

O=C(ONc1ccc(-c2ccccc2)cc1)C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.49
HDAC6 Q9UBN7 6/20 0.49
HDAC2 Q92769 6/20 0.49
HDAC7 Q8WUI4 5/20 0.49
HDAC8 Q9BY41 5/20 0.49
HDAC3 O15379 4/20 0.49
HDAC4 P56524 4/20 0.49
HDAC10 Q969S8 4/20 0.49
HDAC11 Q96DB2 4/20 0.49
HDAC9 Q9UKV0 4/20 0.49
HDAC5 Q9UQL6 4/20 0.49
PTPN1 P18031 3/20 0.44
PTPN11 Q06124 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
TP53 P04637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4832864 0.89 HDAC1 (0.44) HDAC1HDAC6HDAC2HDAC7HDAC8
SCHEMBL1844466 0.76 SMN1; SMN2 (0.50) NPC1RAB9AKMT2AMEN1TP53
SCHEMBL7734069 0.76 LMNA (0.46) HDAC1HDAC6HDAC2HDAC7HDAC8
SCHEMBL27795033 0.74 MMP1 (0.49) KMT2AMEN1HTTMAPT
SCHEMBL13842150 0.73 PTPN1 (0.47) PTPN1PTPN11NPC1RAB9AALDH1A1
SCHEMBL9543659 0.73 HDAC1 (0.50) HDAC1HDAC6HDAC2HDAC7HDAC8
SCHEMBL8755361 0.73 RAB9A (0.71) HDAC1HDAC6HDAC2HDAC7HDAC8
SCHEMBL6028396 0.72 ALDH1A1 (0.57) HDAC1HDAC6HDAC2HDAC7HDAC8
SCHEMBL5716690 0.72 KIF11 (0.45) HDAC1HDAC6HDAC2HDAC7HDAC8
SCHEMBL28148996 0.71 ALDH1A1 (0.45) NPC1RAB9AKMT2ATP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003035615-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-05-01 WO claimed
WO-2003035615-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-05-01 WO disclosed