SCHEMBL7073697

SCHEMBL7073697

COc1ccc2[nH]c(C(=O)O)c([C@@H]3C[C@H]3C(=O)O)c2c1Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CA12 O43570 1/20 0.37
MAPT P10636 1/20 0.36
MDM2 Q00987 6/20 0.36
POLB P06746 1/20 0.35
LMNA P02545 3/20 0.35
KDM4A O75164 1/20 0.34
KDM5A P29375 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
LTC4S Q16873 1/20 0.34
CCR2 P41597 2/20 0.34
CDK8 P49336 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.33
GAA P10253 1/20 0.33
CRHBP P24387 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074273 0.80 MDM2 (0.40) MDM2KDM4AKDM5AKDM5B
SCHEMBL5503145 0.77 PTPN5 (0.37) CA1CA2CA9CA12POLB
SCHEMBL7072708 0.67 GPR17 (0.61) MAPTMDM2POLBCCR2MEN1
SCHEMBL7842628 0.64 KDM4E (0.47) MAPTMDM2POLB
SCHEMBL7817673 0.64 MCL1 (0.48)
SCHEMBL6996736 0.62 ALDH1A1 (0.52) CA1CA2CA9CA12MEN1
SCHEMBL6996735 0.62 ALDH1A1 (0.52) CA1CA2CA9CA12MEN1
SCHEMBL6302418 0.62 ABCB11 (0.55) MAPTLMNACCR2MEN1KMT2A
SCHEMBL6302422 0.62 ABCB11 (0.55) MAPTLMNACCR2MEN1KMT2A
SCHEMBL6594503 0.62 MAPT (0.47) MAPTPOLBLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003504-B1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2003-07-02 EP disclosed