SCHEMBL7075403

SCHEMBL7075403

Cc1nc(-c2ccc(C(=O)N3CCN(C(=O)COc4ccccc4)CC3)cc2)no1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
NPC1 O15118 2/20 0.56
RAB9A P51151 1/20 0.56
MGLL Q99685 1/20 0.55
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
HTT P42858 1/20 0.54
POLB P06746 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
DGAT1 O75907 1/20 0.51
CPT1A P50416 3/20 0.49
CPT2 P23786 2/20 0.49
KDM4E B2RXH2 2/20 0.49
PKM P14618 1/20 0.49
CPT1B Q92523 1/20 0.48
TPSAB1 Q15661 1/20 0.48
TPSD1 Q9BZJ3 1/20 0.48
TPSG1 Q9NRR2 1/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074772 0.84 MGLL (0.66) ALDH1A1MGLLMEN1KMT2APOLB
SCHEMBL7076687 0.80 TSHR (0.59) ALDH1A1NPC1RAB9AMGLLMEN1
SCHEMBL7070548 0.78 MGLL (0.56) ALDH1A1MGLLMEN1KMT2ASMN1; SMN2
SCHEMBL7649408 0.78 DGAT1 (0.58) ALDH1A1MGLLPOLBDGAT1KDM4E
SCHEMBL7075122 0.77 LMNA (0.65) ALDH1A1MGLLHTTSMN1; SMN2
SCHEMBL7073717 0.76 TSHR (0.57) ALDH1A1RAB9AMGLLKMT2ASMN1; SMN2
SCHEMBL7074046 0.76 HDAC4 (0.57) RAB9AMGLL
SCHEMBL7074241 0.76 HDAC4 (0.53) NPC1RAB9AMGLLHTTPOLB
SCHEMBL7076841 0.76 MGLL (0.54) ALDH1A1NPC1RAB9AMGLLHTT
SCHEMBL7071696 0.75 ALDH1A1 (0.61) ALDH1A1NPC1RAB9AMGLLMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed