SCHEMBL4880583

SCHEMBL4880583

COC(=O)c1ccccc1CS(N)(=O)=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA5A P35218 1/20 0.58
CA9 Q16790 1/20 0.58
ALDH1A1 P00352 3/20 0.55
LMNA P02545 2/20 0.55
TSHR P16473 1/20 0.53
HSD17B10 Q99714 2/20 0.51
CFTR P13569 1/20 0.51
HIF1A Q16665 1/20 0.47
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 2/20 0.46
POLB P06746 2/20 0.46
ATM Q13315 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
GLA P06280 1/20 0.44
HTT P42858 1/20 0.43
EGFR P00533 1/20 0.43
NOX4 Q9NPH5 1/20 0.43
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15461583 0.85 ALDH1A1 (0.57) CA1CA2CA5ACA9ALDH1A1
SCHEMBL7363401 0.85 ALDH1A1 (0.57) CA1CA2CA5ACA9ALDH1A1
SCHEMBL9843838 0.84 ALDH1A1 (0.60) CA1CA2CA5ACA9ALDH1A1
SCHEMBL8435579 0.84 TSHR (0.61) CA1CA2CA9ALDH1A1LMNA
SCHEMBL2884550 0.83 ALDH1A1 (0.55) CA1CA2CA5ACA9ALDH1A1
SCHEMBL9843840 0.81 ALDH1A1 (0.57) CA1CA2CA5ACA9ALDH1A1
SCHEMBL10438447 0.81 CA1 (0.44) CA1CA2CA5ACA9ALDH1A1
SCHEMBL4912518 0.81 ALDH1A1 (0.53) CA1CA2CA5ACA9ALDH1A1
SCHEMBL646787 0.81 L3MBTL1 (0.54) CA1CA2CA5ACA9ALDH1A1
SCHEMBL10680197 0.80 KMT2A (0.45) CA1CA2CA5ACA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1171197-A Method for synthesizing herbicide of sulfonylureas ZHANG HUIMING (CN) 1998-01-28 CN claimed
US-H890-H Herbicidal heterocyclicbenzylsulfonamides Rorer, Morris P. (US) 1991-02-05 US claimed
JP-1221366-A None JP disclosed
EP-4276092-A1 COMPOUND LIBRARY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-15 EP disclosed
US-11773058-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2023-10-03 US disclosed
US-11773058-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2023-10-03 US disclosed
US-11773058-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2023-10-03 US disclosed
CN-116783160-A Libraries of compounds 中外制药株式会社 2023-09-19 CN disclosed
EP-3880666-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-06-28 EP disclosed
US-20230024859-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2023-01-26 US disclosed
US-11518739-B2 Sulfonamide carboxamide compounds INFLAZOME LIMITED (IE) 2022-12-06 US disclosed
US-5053072-A HETEROCYCLIC N-ACYLSULFONAMIDES, AND THEIR USE AS HERBICIDES OR GROWTH REGULATORS HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-01 US disclosed
US-H890-H Herbicidal heterocyclicbenzylsulfonamides Rorer, Morris P. (US) 1991-02-05 US disclosed
EP-0353640-A2 Heterocyclic N-acylsulphonamides, process for their preparation, agents containing them and their use as herbicides and plant growth regulators Hoechst Schering AgrEvo GmbH (DE) 1990-02-07 EP disclosed
US-4897105-A (1,2,4)-THIADIAZOLO(2,3-A)PYRIMIDINE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-01-30 US disclosed
JP-H01221366-A PRODUCTION OF SULFONYLUREA DERIVATIVE TAKEDA CHEM IND LTD 1989-09-04 JP disclosed
CN-87102275-A Selective herbicide and manufacturing thereof and use 1988-02-17 CN disclosed
US-4699649-A Herbicidal heterocyclicbenzylsulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-10-13 US disclosed
EP-0239064-A2 Herbicidal compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-09-30 EP disclosed
EP-0164268-A2 Herbicidal sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-12-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230024859-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 CA1 3841/4885CA2 1348/4885CA5A 1703/4885
US-11773058-B2 Sulfonamide carboxamide compounds NLRP3, NOD1, NLRP1 CA1 2065/4885CA2 1651/4885CA5A 1120/4885
US-11518739-B2 Sulfonamide carboxamide compounds NLRP3, PYCARD, NOD1 CA1 2278/4885CA2 1228/4885CA5A 646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.