SCHEMBL7078735

SCHEMBL7078735

NC(=O)c1ccc(NC(=O)C(F)(F)F)c(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP2D6 P10635 1/20 0.49
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MAPK14 Q16539 1/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.38
CYP2C9 P11712 1/20 0.38
PTPN5 P54829 1/20 0.38
VNN1 O95497 1/20 0.38
MAPT P10636 1/20 0.38
XBP1 P17861 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GAA P10253 1/20 0.38
MAOB P27338 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050749 0.84 RAB9A (0.49) RAB9ACYP1A2CYP2C19CYP2D6KMT2A
SCHEMBL6816450 0.81 GAA (0.47) RAB9ACYP1A2CYP2C19CYP2D6KMT2A
SCHEMBL7078236 0.78 CYP1A2 (0.55) RAB9ACYP1A2CYP2C19KMT2ALMNA
SCHEMBL7074254 0.78 ABCC9 (0.53) RAB9ACYP1A2CYP2C19KMT2AMEN1
SCHEMBL16057084 0.76 CA2 (0.59) MAPT
SCHEMBL2709797 0.76 AR (0.45) VNN1MAOB
SCHEMBL28255136 0.75 CYP1A2 (0.59) RAB9ACYP1A2CYP2C19CYP2D6KMT2A
SCHEMBL28148906 0.75 PTGS1 (0.46) RAB9ACYP1A2CYP2C19CYP2D6KMT2A
Hydrochloric Acid SCHEMBL27741712 0.74 AR (0.44) CYP2C19CYP2D6CYP2C9VNN1MAOB
SCHEMBL7079342 0.74 L3MBTL1 (0.60) RAB9ACYP1A2CYP2C19KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030036653-A1 Diaminopyridine-containing thiourea inhibitors of herpes viruses AMERICAN HOME PRODUCTS CORPORATION 2003-02-20 US disclosed
US-20020026055-A1 Aminopyridine-containing thiourea inhibitors of herpes viruses AMERICAN HOME PRODUCTS CORPORATION 2002-02-28 US disclosed
US-20010039348-A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030036653-A1 Diaminopyridine-containing thiourea inhibitors of herpes viruses HAVCR2, CCR6, CXCR6 RAB9A 3069/4885CYP1A2 2695/4885CYP2C19 2905/4885
US-20010039348-A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group CCR6, HAVCR2, BCOR RAB9A 3048/4885CYP1A2 3392/4885CYP2C19 3362/4885
US-20020026055-A1 Aminopyridine-containing thiourea inhibitors of herpes viruses TK1, TPMT, CXCR6 RAB9A 732/4885CYP1A2 3647/4885CYP2C19 1333/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.