SCHEMBL7096791

SCHEMBL7096791

c1ccc(CCCn2cc(-c3ccco3)cn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.48
ADORA1 P30542 9/20 0.48
ADORA2B P29275 6/20 0.47
ADORA3 P0DMS8 6/20 0.47
L3MBTL1 Q9Y468 1/20 0.43
SCD O00767 1/20 0.42
SCD5 Q86SK9 1/20 0.42
SIRT1 Q96EB6 1/20 0.41
FAAH O00519 1/20 0.41
CES1 P23141 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004006 0.83 L3MBTL1 (0.64) ADORA2AADORA1L3MBTL1SCDSCD5
SCHEMBL7092817 0.77 SCD5 (0.45) ADORA2AADORA1ADORA2BADORA3L3MBTL1
SCHEMBL7092854 0.74 HDAC3 (0.49) ADORA2AADORA1ADORA2BADORA3SIRT1
SCHEMBL7098488 0.73 L3MBTL1 (0.57) ADORA2AADORA1ADORA2BADORA3L3MBTL1
SCHEMBL7097845 0.73 ADORA2A (0.43) ADORA2AADORA1ADORA2BADORA3L3MBTL1
SCHEMBL6528550 0.72 SIGMAR1 (0.44) ADORA2AADORA1ADORA2BL3MBTL1
SCHEMBL31224806 0.72 MAOB (0.47) ADORA2AADORA1ADORA2BL3MBTL1
SCHEMBL7096885 0.71 ADORA2A (0.52) ADORA2AADORA1ADORA2BADORA3L3MBTL1
SCHEMBL6690784 0.71 ADORA2A (0.50) ADORA2AADORA1ADORA2BADORA3L3MBTL1
SCHEMBL15014142 0.71 ADORA2A (0.46) ADORA2AADORA1ADORA2BL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed