SCHEMBL710306

SCHEMBL710306

OCc1ccc(Cl)cc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.46
MAPT P10636 2/20 0.41
IDO1 P14902 6/20 0.40
CYP3A4 P08684 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HIF1A Q16665 2/20 0.40
HTT P42858 2/20 0.40
MEN1 O00255 1/20 0.40
SLC22A1 O15245 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSPD1 P10809 1/20 0.40
HSPA5 P11021 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
ALOX12 P18054 1/20 0.40
CASP1 P29466 1/20 0.40
BLM P54132 1/20 0.40
HSPE1 P61604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30749355 1.00 PYCR1 (0.46) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL3634811 0.83 PYCR1 (0.44) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL500015 0.82 CYP3A4 (0.45) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL17410220 0.79 PYCR1 (0.41) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL597241 0.79 MAOA (0.41) MAPTHTTMEN1KMT2APSEN1
SCHEMBL596499 0.79 MAOA (0.41) LMNAPPARASLC6A4
SCHEMBL29485890 0.79 PYCR1 (0.47) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL26078400 0.79 PYCR1 (0.47) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL979069 0.79 PYCR1 (0.47) PYCR1MAPTIDO1CYP3A4SMN1; SMN2
SCHEMBL29493203 0.78 IDO1 (0.50) MAPTIDO1CYP3A4SMN1; SMN2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 208 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160977-A2 BIPHENYL AMIDES WITH MODIFIED ETHER GROUPS AS HSP90 INHIBITORS AND HSP70 INDUCERS The University of Kansas (US) 2017-05-03 EP claimed
WO-2015200514-A2 BIPHENYL AMIDES WITH MODIFIED ETHER GROUPS AS HSP90 INHIBITORS AND HSP70 INDUCERS THE UNIVERSITY OF KANSAS (US) 2015-12-30 WO claimed
US-12459950-B2 Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) PRELUDE THERAPEUTICS, INCORPORATED (US) 2025-11-04 US disclosed
US-12440506-B2 Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) PRELUDE THERAPEUTICS, INCORPORATED (US) 2025-10-14 US disclosed
EP-4573096-A1 INHIBITORS OF MYELOPEROXIDASE Astrazeneca AB (SE) 2025-06-25 EP disclosed
CN-119894896-A Inhibitors of green peroxidase 阿斯利康(瑞典)有限公司 2025-04-25 CN disclosed
US-20240343740-A1 MACROCYCLIC GLUCAGON-LIKE PEPTIDE 1 RECEPTOR AGONISTS ELI LILLY AND COMPANY 2024-10-17 US disclosed
US-20240166642-A1 INHIBITORS OF MYELOPEROXIDASE ASTRAZENECA AB (SE) 2024-05-23 US disclosed
EP-4341255-A1 MACROCYCLIC GLUCAGON-LIKE PEPTIDE 1 RECEPTOR AGONISTS Eli Lilly and Company (US) 2024-03-27 EP disclosed
WO-2024038131-A1 INHIBITORS OF MYELOPEROXIDASE ASTRAZENECA AB (SE) 2024-02-22 WO disclosed
CN-117355517-A Macrocyclic glucagon-like peptide 1 receptor agonists 伊莱利利公司 2024-01-05 CN disclosed
WO-2010055005-A1 NAPHTHYLACETIC ACIDS F. HOFFMANN-LA ROCHE AG (CH) 2010-05-20 WO disclosed
WO-2009158426-A1 6-SUBSTITUTED PHENOXYCHROMAN CARBOXYLIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2009-12-30 WO disclosed
EP-1805165-B1 1-(HETERO)ARYL-3-AMINO-PYRROLIDINE DERIVATIVES FOR USE AS MGLUR3 RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2009-12-16 EP disclosed
US-20080300266-A1 1-(Hetero)Aryl-3-Amino-Pyrrolidine Derivatives for Use as Mglur3 Antagonists ELI LILLY AND COMPANY (US) 2008-12-04 US disclosed
CN-101094846-A 1- (hetero) aryl-3-amino-pyrrolidine derivatives as MGLUR3 receptor antagonists LILLY CO ELI (US) 2007-12-26 CN disclosed
EP-1805165-A1 1-(HETERO)ARYL-3-AMINO-PYROLLIDINE DERIVATIVES FOR USE AS MGLUR3 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2007-07-11 EP disclosed
WO-2006044454-A1 1-(HETERO)ARYL-3-AMINO-PYROLLIDINE DERIVATIVES FOR USE AS MGLUR3 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2006-04-27 WO disclosed
US-3985889-A 1,3-DIHYDROSPIRO(ISOBENZOFURAN); ANALGETIC AGENTS AMERICAN HOECHST CORPORATION (US) 1976-10-12 US disclosed
US-3962259-A TRANQUILIZERS, ANALGETIC AGENTS AMERICAN HOECHST CORPORATION (US) 1976-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240343740-A1 MACROCYCLIC GLUCAGON-LIKE PEPTIDE 1 RECEPTOR AGONISTS GLP1R, GCGR, GIPR PYCR1 1751/4885MAPT 4616/4885IDO1 3650/4885
US-12459950-B2 Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) PRMT5, PRMT1, PRMT6 PYCR1 2973/4885MAPT 1314/4885IDO1 2912/4885
US-20240166642-A1 INHIBITORS OF MYELOPEROXIDASE MPO, XDH, EPX PYCR1 207/4885MAPT 3935/4885IDO1 544/4885
US-12440506-B2 Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) PRMT5, PRMT1, PRMT6 PYCR1 2561/4885MAPT 2168/4885IDO1 2534/4885
US-20080300266-A1 1-(Hetero)Aryl-3-Amino-Pyrrolidine Derivatives for Use as Mglur3 Antagonists GRM3, GRM1, GRIA3 PYCR1 665/4885MAPT 2322/4885IDO1 1072/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.