SCHEMBL7145208

SCHEMBL7145208

CC(C)(C)OC(=O)c1cccc2nc(CCl)[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.38
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
MEN1 O00255 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
KMT2A Q03164 2/20 0.35
GAA P10253 2/20 0.35
PKM P14618 1/20 0.35
PTPN1 P18031 1/20 0.35
KDM4E B2RXH2 4/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
GLA P06280 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002080 0.85 KDM4E (0.48) MEN1NPC1RAB9AKMT2AGAA
SCHEMBL2340375 0.84 ADRA1A (0.37) BCHEADRA1AADRA1BMEN1NPC1
SCHEMBL938871 0.80 BCHE (0.44) BCHEACACBACACAMEN1NPC1
SCHEMBL4033463 0.80 PARP1 (0.43) KDM4EHPGD
SCHEMBL4713440 0.79 TSHR (0.52) ADRA1AADRA1BNPC1RAB9AKDM4E
SCHEMBL7003014 0.78 PLK4 (0.45) RAB9AKDM4ERECQLSMN1; SMN2HSD17B10
SCHEMBL5886053 0.77 TNKS (0.43) NPC1RAB9AKMT2AGAAPKM
SCHEMBL11947879 0.76 CACNA1G (0.44) BCHEMEN1NPC1RAB9AKMT2A
SCHEMBL7721019 0.73 DDAH1 (0.44) MEN1KMT2AGAAKDM4EALDH1A1
SCHEMBL19488865 0.72 LMNA (0.37) MEN1KMT2AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1237061-C Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2006-01-18 CN disclosed
CN-1458929-A Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2003-11-26 CN disclosed
EP-1317451-A1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2003-06-11 EP disclosed
WO-2002034745-A1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC. (CA) 2002-05-02 WO disclosed
WO-1999011612-A2 SUBSTITUTED CYCLIC COMPOUNDS AND MIXTURES COMPRISING SAME ISIS PHARMACEUTICALS, INC. (US) 1999-03-11 WO disclosed