Predicted protein targets (top 16)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | PTGDR2 | Q9Y5Y4 | 12/20 | 0.54 |
| ▸ | ATP4A | P20648 | 2/20 | 0.48 |
| ▸ | ATP4B | P51164 | 2/20 | 0.48 |
| ▸ | KDM4E | B2RXH2 | 4/20 | 0.47 |
| ▸ | POLB | P06746 | 1/20 | 0.47 |
| ▸ | ALDH1A1 | P00352 | 4/20 | 0.46 |
| ▸ | MAPT | P10636 | 2/20 | 0.46 |
| ▸ | GLA | P06280 | 2/20 | 0.45 |
| ▸ | CYP1A2 | P05177 | 1/20 | 0.44 |
| ▸ | CYP2C9 | P11712 | 1/20 | 0.44 |
| ▸ | HPGD | P15428 | 1/20 | 0.44 |
| ▸ | CYP2C19 | P33261 | 1/20 | 0.44 |
| ▸ | NPC1 | O15118 | 1/20 | 0.44 |
| ▸ | LMNA | P02545 | 1/20 | 0.44 |
| ▸ | GAA | P10253 | 1/20 | 0.44 |
| ▸ | RAB9A | P51151 | 1/20 | 0.44 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL15130547 | 0.83 | RAB9A (0.44) | PTGDR2KDM4EALDH1A1MAPTGLA | |
| SCHEMBL11466220 | 0.82 | ALDH1A1 (0.67) | PTGDR2ATP4AATP4BKDM4EPOLB | |
| SCHEMBL8005690 | 0.80 | PTGDR2 (0.68) | PTGDR2ATP4AATP4BKDM4ECYP1A2 | |
| SCHEMBL11100736 | 0.73 | PTGDR2 (0.82) | PTGDR2KDM4EPOLBALDH1A1MAPT | |
| SCHEMBL11097514 | 0.72 | PTGDR2 (0.64) | PTGDR2KDM4EPOLBALDH1A1MAPT | |
| SCHEMBL28167586 | 0.71 | ALOX5 (0.43) | KDM4EALDH1A1MAPTGLANPC1 | |
| SCHEMBL10662994 | 0.70 | ATP4A (0.73) | PTGDR2ATP4AATP4BALDH1A1MAPT | |
| SCHEMBL9628554 | 0.70 | TRPM8 (0.62) | PTGDR2MAPT | |
| SCHEMBL23424392 | 0.70 | PTGDR2 (0.52) | PTGDR2KDM4EALDH1A1MAPTHPGD | |
| SCHEMBL14840398 | 0.69 | CDC7 (0.55) | MAPT |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-9273115-B2 | Method for controlling the biological activity of a protein in a vertebrate cell | CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) | 2016-03-01 | — | — | US | claimed |
| EP-2389391-B1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | CENTRE NAT RECH SCIENT (FR) | 2014-03-12 | — | — | EP | claimed |
| US-20120052570-A1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) | 2012-03-01 | — | — | US | claimed |
| EP-2389391-A1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | Centre National De La Recherche Scientifique CNRS (FR) | 2011-11-30 | — | — | EP | claimed |
| US-20110255621-A1 | SYNCHRONIZED MULTIPOINT-TO-POINT COMMUNICATION USING ORTHOGONAL FREQUENCY DIVISION | HTC CORPORATION | 2011-10-20 | — | — | US | claimed |
| WO-2010084171-A1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) | 2010-07-29 | — | — | WO | claimed |
| US-9273115-B2 | Method for controlling the biological activity of a protein in a vertebrate cell | CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) | 2016-03-01 | — | — | US | disclosed |
| EP-2389391-B1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | CENTRE NAT RECH SCIENT (FR) | 2014-03-12 | — | — | EP | disclosed |
| US-20120052570-A1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) | 2012-03-01 | — | — | US | disclosed |
| EP-2389391-A1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | Centre National De La Recherche Scientifique CNRS (FR) | 2011-11-30 | — | — | EP | disclosed |
| US-20110255621-A1 | SYNCHRONIZED MULTIPOINT-TO-POINT COMMUNICATION USING ORTHOGONAL FREQUENCY DIVISION | HTC CORPORATION | 2011-10-20 | — | — | US | disclosed |
| WO-2010084171-A1 | METHOD FOR TEMPORALLY CONTROLLING THE BIOLOGICAL ACTIVITY OF PROTEINS IN VERTEBRATES, AND APPLICATIONS THEREOF | CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) | 2010-07-29 | — | — | WO | disclosed |
| US-20060199250-A1 | Method for generating a mutant protein which efficiently binds a target molecule | BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS, THE | 2006-09-07 | — | — | US | disclosed |
| WO-2000019994-A9 | ESTROGEN RECEPTOR LIGANDS | UNIV ILLINOIS (US) | 2000-08-31 | — | — | WO | disclosed |
| WO-2000019994-A1 | ESTROGEN RECEPTOR LIGANDS | BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) | 2000-04-13 | — | — | WO | disclosed |