SCHEMBL7196066

SCHEMBL7196066

COCOc1ccc(-c2[nH]c3cc(Cl)c(F)cc3c(=O)c2C(=O)OC)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 5/20 0.38
PRKAG1 P54619 5/20 0.38
PRKAA2 P54646 5/20 0.38
PRKAA1 Q13131 5/20 0.38
PRKAG3 Q9UGI9 5/20 0.38
PRKAG2 Q9UGJ0 5/20 0.38
PRKAB1 Q9Y478 5/20 0.38
ALOX5 P09917 1/20 0.36
NPC1 O15118 1/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 1/20 0.36
NR4A2 P43354 1/20 0.36
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
IMPDH2 P12268 1/20 0.35
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008377 0.91 PRKAB2 (0.42) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL25234089 0.73 ALOX5 (0.47) ALOX5NPC1KDM4ENR4A2MAPT
SCHEMBL7009049 0.73 ALDH1A1 (0.42) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL25197469 0.72 NR4A2 (0.51) ALOX5NR4A2
SCHEMBL7016620 0.71 KIF11 (0.42) NPC1KDM4E
SCHEMBL25200108 0.69 ALOX5 (0.49) ALOX5KDM4ENR4A2MAPTTP53
SCHEMBL25212344 0.69 NR4A2 (0.52) ALOX5NR4A2
SCHEMBL31312623 0.68 TUBB4A (0.47) ALOX5KDM4EGAANR4A2MAPT
SCHEMBL10478188 0.67 NR4A2 (0.53) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL7010787 0.67 ALOX5 (0.56) ALOX5NPC1KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313708-A1 QUINOLINE ANTIBACTERIAL COMPOUNDS AND METHODS OF USE THEREOF CHIRON CORPORATION (US) 2003-05-28 EP disclosed
WO-2002018345-A1 QUINOLINE ANTIBACTERIAL COMPOUNDS AND METHODS OF USE THEREOF CHIRON CORPORATION (US) 2002-03-07 WO disclosed