SCHEMBL7009049

SCHEMBL7009049

COCOc1ccc(-c2[nH]c3cc(N4CCN(C)CC4)c(F)cc3c(=O)c2C(=O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
DRD3 P35462 1/20 0.42
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
LMNA P02545 3/20 0.40
KDM4E B2RXH2 5/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
KIF11 P52732 4/20 0.38
GAA P10253 1/20 0.36
RAD52 P43351 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CG P48736 1/20 0.36
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016620 0.88 KIF11 (0.42) ALDH1A1KMT2AMEN1LMNAKDM4E
SCHEMBL7008377 0.81 PRKAB2 (0.42) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL7014803 0.76 KIF11 (0.52) ALDH1A1DRD3KMT2AMEN1LMNA
SCHEMBL11204174 0.74 ALDH1A1 (0.47) ALDH1A1DRD3KMT2AMEN1LMNA
SCHEMBL7015614 0.74 LMNA (0.75) ALDH1A1DRD3KMT2AMEN1LMNA
SCHEMBL7196066 0.73 PRKAB2 (0.38) KDM4ENPC1GAAPRKAB2PRKAG1
SCHEMBL7013585 0.71 KDM4E (0.42) ALDH1A1KMT2AMEN1LMNAKDM4E
SCHEMBL7011748 0.70 ALOX5 (0.46) ALDH1A1KMT2AMEN1LMNAKDM4E
SCHEMBL9379704 0.69 ALDH1A1 (0.58) ALDH1A1DRD3KMT2AMEN1LMNA
SCHEMBL11208613 0.68 GAA (0.47) ALDH1A1DRD3KMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313708-A1 QUINOLINE ANTIBACTERIAL COMPOUNDS AND METHODS OF USE THEREOF CHIRON CORPORATION (US) 2003-05-28 EP disclosed
WO-2002018345-A1 QUINOLINE ANTIBACTERIAL COMPOUNDS AND METHODS OF USE THEREOF CHIRON CORPORATION (US) 2002-03-07 WO disclosed