SCHEMBL7212138

SCHEMBL7212138

CCCC(C(C)C(=O)O)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 9/20 0.54
MMP9 P14780 6/20 0.54
MMP1 P03956 11/20 0.54
MMP2 P08253 9/20 0.54
MMP3 P08254 8/20 0.54
PDE4A P27815 3/20 0.54
PDE4B Q07343 3/20 0.54
PDE4C Q08493 3/20 0.54
PDE4D Q08499 3/20 0.54
ADAM17 P78536 2/20 0.52
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KEAP1 Q14145 2/20 0.44
NFE2L2 Q16236 1/20 0.44
MMP8 P22894 1/20 0.44
MMP12 P39900 1/20 0.44
MMP14 P50281 1/20 0.44
MMP16 P51512 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7207041 0.91 MMP1 (0.61) MMP13MMP9MMP1MMP2MMP3
SCHEMBL7207035 0.79 MMP1 (0.54) MMP13MMP9MMP1MMP2MMP3
SCHEMBL6933212 0.76 MMP13 (0.74) MMP13MMP9MMP1MMP2MMP3
SCHEMBL13043584 0.76 MMP1 (0.85) MMP13MMP9MMP1MMP2MMP3
SCHEMBL7352846 0.76 MMP13 (0.60) MMP13MMP9MMP1MMP2MMP3
SCHEMBL7306444 0.74 MMP1 (0.65) MMP13MMP9MMP1MMP2MMP3
SCHEMBL7346604 0.74 MMP13 (0.75) MMP13MMP9MMP1MMP2MMP3
SCHEMBL6928909 0.74 MMP13 (0.75) MMP13MMP9MMP1MMP2MMP3
Hydroxyamine SCHEMBL8224643 0.74 PDE4A (0.50) MMP13MMP9MMP1MMP2MMP3
SCHEMBL7077429 0.73 HTT (0.52) MMP13MMP9MMP1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed